Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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2,506
Tocris Bioscience™ XAP 044
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective mGlu7 antagonist
| Inhibitors | XAP 044 |
|---|---|
| Product Type | XAP 044 |
| Molecular Weight (g/mol) | 380.13 |
| Purity | >98% |
2,507
Tocris Bioscience™ SU 5416
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CAS: 204005-46-9 Molecular Formula: C15H14N2O
| CAS | 204005-46-9 |
|---|---|
| Molecular Formula | C15H14N2O |
2,508
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Tocris Bioscience™ FTY 720
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Tocris Bioscience™ FTY 720
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent S1P receptor agonist; also immunosuppressant
| Target | Sphingosine-1-phosphate Receptor |
|---|---|
| CAS | 162359-56-0 |
| Product Type | Agonist |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H33NO2.HCl |
| Formula Weight | 343.93g/mol |
2,509
Tocris Bioscience™ AZ 628
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CAS: 878739-06-1 Molecular Formula: C27H25N5O2
| CAS | 878739-06-1 |
|---|---|
| Molecular Formula | C27H25N5O2 |
2,510
Tocris Bioscience™ CNQX disodium salt
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CAS: 479347-85-8 Molecular Formula: C9H2N4Na2O4
| CAS | 479347-85-8 |
|---|---|
| Molecular Formula | C9H2N4Na2O4 |
2,511
Tocris Bioscience™ SGC SMARCA-BRDVIII
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Potent and selective SMARCA2/4 and PB1(bromo 5)-selective SWI/SNF bromodomain inhibitor
| Target | Bromodomain Inhibitors |
|---|---|
| CAS | 1997319-84-2 |
| Purity | 0.98 |
| Chemical Name or Material | 1,1-Dimethylethyl 4-[3-amino-6-(2-hydroxyphenyl)-4-pyridazinyl]-1-piperazinecarboxylate bromodomains |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H25N5O3 |
2,512
Tocris Bioscience™ 25-Hydroxycholesterol
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Antiviral; also α-crystallin (cryAB) chaperone
2,513
Tocris Bioscience™ BI-6901
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Potent and selective CCR10 antagonist
2,514
Tocris Bioscience™ EN6
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H+ ATPase activator; activates autophagy; inactivates mTORC1 signaling
| Target | H+-ATPase Inhibitors |
|---|---|
| CAS | 1808714-73-9 |
| Purity | 0.98 |
| Chemical Name or Material | N-[4-Fluoro-3-[(1-oxo-2-propen-1-yl)amino]phenyl]-1-(2-fluorophenyl)-1 H-pyrazole-4-carboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H14F2N4O2 |
2,515
Tocris Bioscience™ Ro 64-5229
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 246852-46-0 Molecular Formula: C17H19Cl2N3O
| CAS | 246852-46-0 |
|---|---|
| Molecular Formula | C17H19Cl2N3O |
2,516
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Tocris Bioscience™ CP 690550 citrate
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Tocris Bioscience™ CP 690550 citrate
Greener Choice
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CAS: 540737-29-9 Molecular Formula: C22H28N6O8
| CAS | 540737-29-9 |
|---|---|
| Molecular Formula | C22H28N6O8 |
2,517
Tocris Bioscience™ Perifosine
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PKB/Akt inhibitor; also modulates Kv2.1 current
| CAS | 157716-52-4 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Color | White |
| Solubility | Soluble to 100mM in water and to 100mM in ethanol |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | Perifosine |
| Recommended Storage | Store at -20°C |
| Synonym | Octadecyl-(1,1-dimethyl-4-piperidylio) phosphate |
| Molecular Formula | C25H52NO4P |
| Formula Weight | 461.66 |
2,518
Tocris Bioscience™ CCCP
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CAS: 555-60-2 Molecular Formula: C9H5ClN4
| CAS | 555-60-2 |
|---|---|
| Molecular Formula | C9H5ClN4 |
2,519
Tocris Bioscience™ Balicatib
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Potent and selective cathepsin K inhibitor
| Target | Synthetic Cathepsin Inhibitors |
|---|---|
| CAS | 354813-19-7 |
| Purity | >98% |
| Chemical Name or Material | N-[1-(Cyanomethylcarbamoyl)cyclohexyl]-4-(4-propylpiperazin-1-yl)benzamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C23H33N5O2 |
| Formula Weight | 411.54 |
2,520
Tocris Bioscience™ SB 271046 hydrochloride
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CAS: 209481-20-9 Molecular Formula: C20H23Cl2N3O3S2
| CAS | 209481-20-9 |
|---|---|
| Molecular Formula | C20H23Cl2N3O3S2 |